Description

CAS № 2894-68-0
Purity ≥98%
Synonyms:2′-Chlorodiazepam;Ro 5-3448

Diazepam is a benzodiazepine drug that produces psychoactive effects by enhancing signaling through the γ-aminobutyric acid (GABA) receptor GABAA.1 Diclazepam is a 2’-chloro derivative of diazepam that has emerged as a designer drug.2 It is metabolized in vivo into the pharmacologically active benzodiazepines delorazepam, lorazepam, and lormetazepam, which can be detected in urine for 6, 19, and 11 days, respectively.2 The product is intended for forensic and research applications.Currently, the drug is sold as a research chemical and not yet marketed as a medication because it has not been tested systematically in humans. Diclazepam’s closest relatives and two main metabolites are delorazepam and lormetazepam. Deloraepam has around 10 times the potency value of diazepam and lorometazepam has a potency of around 10 to 12 times of delorazepam.